studies established

Psychedelic effects of psilocybin correlate with serotonin 2A receptor occupancy and plasma psilocin levels

The intensity of the subjective psychedelic experience tracked directly with 5-HT2A receptor occupancy and blood psilocin levels, confirming the receptor mechanism in living humans.

Madsen, Fisher, Burmester, et al. January 1, 2019

Key finding — The intensity of the subjective psychedelic experience tracked directly with 5-HT2A receptor occupancy and blood psilocin levels, confirming the receptor mechanism in living humans.

Study at a glance

FieldDetail
InstitutionUniversity of Copenhagen
DesignWithin-subject pharmacology and PET study
Sample size8 participants
InterventionOral psilocybin with PET imaging and plasma sampling
Year2019
ConditionHealthy volunteers (pharmacology)
JournalNeuropsychopharmacology
Evidenceestablished

Limitations

Very small sample; PET occupancy modeling involves assumptions, and healthy volunteers may differ from clinical populations.

Editorial note

A mechanistic study that directly linked the felt intensity of a psilocybin experience to receptor occupancy and drug levels in the body — closing part of the gap between molecule and experience.

Read the primary source →


Summary written by MMI Editorial for clarity. Always consult the primary source for full methodology and results. The confidence rating reflects our assessment of evidence strength.